SCHEMBL9002064

SCHEMBL9002064

CC(COc1cccc2nccn12)NS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 10/20 0.42
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
HTR6 P50406 1/20 0.37
EDNRA P25101 2/20 0.37
HCRTR1 O43613 1/20 0.36
SLC6A9 P48067 3/20 0.36
EDNRB P24530 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SCN1A P35498 1/20 0.35
SCN2A Q99250 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SCN3A Q9NY46 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002378 0.84 NR3C1 (0.38) NR3C1ALDH1A1
SCHEMBL9002438 0.82 CYP3A4 (0.46) SLC6A9KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9002369 0.81 CYP3A4 (0.50) HTR6KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9002497 0.79 ALDH1A1 (0.54) HTR6KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL20025843 0.72 SLC1A3 (0.55) SLC1A3SLC1A2SLC1A1EDNRAHCRTR1
SCHEMBL9001942 0.70 CYP3A4 (0.45) HTR6SLC6A9KDM4EALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9001969 0.69 SCN1A (0.46) HTR6SLC6A9KDM4EALDH1A1CYP1A2
SCHEMBL13951132 0.69 SLC1A3 (0.54) SLC1A3SLC1A2SLC1A1EDNRAHCRTR1
SCHEMBL12132457 0.69 KDM4E (0.56) SLC1A3SLC1A2SLC1A1EDNRAHCRTR1
SCHEMBL9001901 0.69 CYP3A4 (0.48) HTR6KDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed