SCHEMBL9002369

SCHEMBL9002369

O=S(=O)(NCCCOc1cccc2nccn12)c1cccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
SCN1A P35498 2/20 0.50
SCN2A Q99250 2/20 0.50
SCN3A Q9NY46 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NPY5R Q15761 5/20 0.44
HTR7 P34969 4/20 0.44
AGTR1 P30556 1/20 0.44
AGTR2 P50052 1/20 0.44
HTR6 P50406 2/20 0.41
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
MEN1 O00255 2/20 0.41
PRKD3 O94806 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002438 0.97 CYP3A4 (0.46) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9002497 0.96 ALDH1A1 (0.54) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9002415 0.83 MAPK1 (0.51) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL9001901 0.81 CYP3A4 (0.48) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9002064 0.81 NR3C1 (0.42) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9002030 0.81 CYP3A4 (0.50) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9001991 0.79 POLB (0.38) KDM4EALDH1A1NPY5RMEN1PRKD3
SCHEMBL9001942 0.79 CYP3A4 (0.45) CYP3A4SCN1ASCN2ASCN3AKDM4E
Hydrochloric Acid SCHEMBL9001969 0.78 SCN1A (0.46) CYP3A4SCN1ASCN2ASCN3AKDM4E
SCHEMBL9001957 0.77 IDO1 (0.43) NPY5RMEN1KMT2APRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed