SCHEMBL9002188

SCHEMBL9002188

CCOc1ccc(CC(CO)NC(=O)OCc2ccccc2)cc1Br

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 3/20 0.50
CTRB1 P17538 2/20 0.50
MEN1 O00255 2/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
CYP3A4 P08684 5/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
TSHR P16473 2/20 0.44
SYK P43405 1/20 0.43
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002209 0.89 KMT2A (0.48) ALDH1A1KMT2ACTRB1MEN1LMNA
SCHEMBL9001816 0.88 CTRB1 (0.50) ALDH1A1KMT2ACTRB1MEN1SMN1; SMN2
SCHEMBL9002042 0.86 KMT2A (0.46) ALDH1A1KMT2ACTRB1MEN1LMNA
SCHEMBL9001915 0.86 SMN1; SMN2 (0.46) ALDH1A1KMT2ACTRB1MEN1LMNA
SCHEMBL8612085 0.82 CTRB1 (0.60) ALDH1A1CTRB1MAPTSMN1; SMN2CYP3A4
SCHEMBL8612079 0.82 CTRB1 (0.60) ALDH1A1CTRB1MAPTSMN1; SMN2CYP3A4
SCHEMBL8668738 0.81 CTRB1 (0.52) ALDH1A1KMT2ACTRB1MEN1SMN1; SMN2
SCHEMBL3989318 0.79 CTRB1 (0.50) ALDH1A1KMT2ACTRB1MEN1SMN1; SMN2
SCHEMBL2435512 0.79 CTRB1 (0.76) ALDH1A1CTRB1SMN1; SMN2CYP3A4CYP1A2
SCHEMBL1051352 0.79 CTRB1 (0.76) ALDH1A1CTRB1SMN1; SMN2CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731784-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-18 EP disclosed
WO-1995015306-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed