SCHEMBL9002209

SCHEMBL9002209

CCOc1ccc(CC(COC(C)=O)NC(=O)OCc2ccccc2)cc1Br

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
CTRB1 P17538 2/20 0.47
ALDH1A1 P00352 4/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
SYK P43405 1/20 0.41
CYP3A4 P08684 1/20 0.41
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002188 0.89 ALDH1A1 (0.50) KMT2AMEN1CTRB1ALDH1A1LMNA
SCHEMBL9002042 0.88 KMT2A (0.46) KMT2AMEN1CTRB1ALDH1A1LMNA
SCHEMBL9001915 0.83 SMN1; SMN2 (0.46) KMT2AMEN1CTRB1ALDH1A1LMNA
SCHEMBL9810151 0.77 SYK (0.60) KMT2AMEN1CTRB1ALDH1A1LMNA
SCHEMBL9001816 0.77 CTRB1 (0.50) KMT2AMEN1CTRB1ALDH1A1SMN1; SMN2
SCHEMBL10332296 0.73 SYK (0.61) KMT2AMEN1CTRB1ALDH1A1LMNA
SCHEMBL8612085 0.71 CTRB1 (0.60) CTRB1ALDH1A1MAPTSMN1; SMN2CYP3A4
SCHEMBL8612079 0.71 CTRB1 (0.60) CTRB1ALDH1A1MAPTSMN1; SMN2CYP3A4
SCHEMBL17275393 0.71 CTSS (0.55) CTRB1ALDH1A1CTSLCTSBCTSS
SCHEMBL14595243 0.71 CTRB1 (0.74) CTRB1ALDH1A1SYKCYP3A4CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731784-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-18 EP disclosed
WO-1995015306-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed