SCHEMBL9002291

SCHEMBL9002291

CCCCS(=O)(=O)NCCSc1cccc2nccn12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 1/20 0.34
TBXA2R P21731 1/20 0.33
TBXAS1 P24557 1/20 0.33
AR P10275 1/20 0.32
HSD17B10 Q99714 2/20 0.32
CCR4 P51679 1/20 0.32
CDK8 P49336 2/20 0.32
ROCK1 Q13464 2/20 0.32
FLT1 P17948 1/20 0.32
CDK9 P50750 1/20 0.32
LIMK1 P53667 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
CHEK1 O14757 1/20 0.32
MAP4K4 O95819 1/20 0.32
CSF1R P07333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001931 0.96 KDM4E (0.39) HPGDKDM4EALDH1A1MAPTGAA
SCHEMBL9002012 0.96 KDM4E (0.39) HPGDKDM4EALDH1A1MAPTGAA
SCHEMBL9002373 0.93 KDM4E (0.36) KDM4EALDH1A1MAPTGAATBXAS1
SCHEMBL9002202 0.90 CHEK1 (0.32) ALDH1A1CDK8ROCK1CHEK1MAP4K4
SCHEMBL9002027 0.90 CNR2 (0.36) KDM4EALDH1A1MAPTGAALMNA
SCHEMBL9002172 0.83 MAPT (0.43) ALDH1A1MAPTGAALMNAHSD17B10
Hydrochloric Acid SCHEMBL9001908 0.82 MAPT (0.42) ALDH1A1MAPTGAALMNAHSD17B10
SCHEMBL9002262 0.81 NPY5R (0.33) ALDH1A1MAPTGAAHSD17B10CDK8
SCHEMBL9002013 0.79 POLB (0.37) ALDH1A1MAPTLMNAHSD17B10CDK8
SCHEMBL9002005 0.79 HTT (0.43) HPGDKDM4EALDH1A1GAACDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed