SCHEMBL9003239

SCHEMBL9003239

COC(=O)/C=C/N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2780501 1.00
SCHEMBL427301 1.00
Hydrogen Peroxide SCHEMBL29015874 0.95 NFE2L2 (0.60)
Dimethyl Maleate SCHEMBL75864 0.81 NFE2L2 (1.00)
Dimethyl Fumarate SCHEMBL11668350 0.81 NFE2L2 (1.00)
Dimethyl Fumarate SCHEMBL41836 0.81 NFE2L2 (1.00)
Dimethyl Fumarate SCHEMBL41835 0.81 NFE2L2 (1.00)
Dimethyl Maleate SCHEMBL7057629 0.78 NFE2L2 (0.93)
Dimethyl Maleate SCHEMBL6505431 0.78 NFE2L2 (0.93)
Dimethyl Fumarate SCHEMBL21219085 0.78 NFE2L2 (0.93)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122010831-A Preparation method of 4-trifluoromethyl nicotinic acid 衢州凯沃化工有限公司 2026-05-12 CN claimed
CN-114349694-B Synthetic method of 4-trifluoromethyl nicotinic acid 淮北龙溪生物科技有限公司 2022-11-08 CN claimed
EP-0326389-B1 Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES (JP) 1996-09-11 EP claimed
US-4935516-A Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES, LTD. (JP) 1990-06-19 US claimed
EP-0326389-A2 Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES, LTD. (JP) 1989-08-02 EP claimed
CN-119331364-A Special cable protective sleeve material for truck and preparation method thereof 扬州诺恒特种线缆有限公司 2025-01-21 CN disclosed
CN-117659904-A high-PID-resistance photovoltaic adhesive film and preparation method thereof 江苏景宏新材料科技有限公司 2024-03-08 CN disclosed
CN-115261859-B Copper etching liquid composition and preparation method thereof 李祥庆 2023-06-20 CN disclosed
CN-114349694-B Synthetic method of 4-trifluoromethyl nicotinic acid 淮北龙溪生物科技有限公司 2022-11-08 CN disclosed
CN-115261859-A Copper etching solution composition and preparation method thereof 李祥庆 2022-11-01 CN disclosed
CN-115197651-A Preparation method of Japanese paper account adhesive tape 东莞市玛仕金科技有限公司 2022-10-18 CN disclosed
CN-114349694-A Synthetic method of 4-trifluoromethyl nicotinic acid 淮北龙溪生物科技有限公司 2022-04-15 CN disclosed
EP-2751076-B1 SYNTHESIS METHOD AND INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2018-04-25 EP disclosed
EP-2558445-B1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2017-03-22 EP disclosed
CN-101460198-B Thermosensitive polyphosphazene-bioactive molecule conjugate, preparation method and application thereof KOREA INST SCI & TECH 2013-08-07 CN disclosed
US-7563782-B2 Optically active stereoisomer of efonidipine analogs; R-configuration of the 4-position on dihydropyridine ring; kidney insufficiency; hypercardia; congestive heart failure; cardiomyopathy; arterial sclerosis; antifibrillatory/antiarrhythmia agents; cardiovascular disorders; antiedemic/antiinflammatory NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-07-21 US disclosed
CN-101460198-A Thermosensitive polyphosphazene-bioactive molecule conjugate, preparation method and application thereof KOREA INST SCI & TECH (KR) 2009-06-17 CN disclosed
EP-0326389-B1 Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES (JP) 1996-09-11 EP disclosed
US-4935516-A Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES, LTD. (JP) 1990-06-19 US disclosed
EP-0326389-A2 Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES, LTD. (JP) 1989-08-02 EP disclosed