SCHEMBL900885

SCHEMBL900885

[CH2]c1c(F)cccc1OC(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
POLB P06746 1/20 0.38
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 3/20 0.37
KCNH2 Q12809 2/20 0.37
ALDH1A1 P00352 5/20 0.36
KCNN4 O15554 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 2/20 0.36
DRD1 P21728 1/20 0.35
SLC6A3 Q01959 1/20 0.34
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 2/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
ULK1 O75385 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847783 0.87 ALDH1A1 (0.40) KMT2APOLBALDH1A1SMN1; SMN2HTT
SCHEMBL26617142 0.82 MCHR1 (0.39) KMT2APOLBKCNH2ALDH1A1KCNN4
SCHEMBL23588427 0.78 SLC6A2 (0.48) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL7782409 0.78 KMT2A (0.53) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL900624 0.78 ALDH1A1 (0.49) KMT2APOLBALDH1A1SMN1; SMN2HTT
SCHEMBL21630656 0.75 KMT2A (0.44) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL900886 0.75 KMT2A (0.44) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL16502595 0.75 KMT2A (0.44) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL30719260 0.75 KMT2A (0.44) KMT2APOLBSLC6A2SLC6A4KCNH2
SCHEMBL12474316 0.75 KMT2A (0.37) KMT2APOLBSLC6A2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3837250-A1 PYRAZINE COMPOUNDS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD (CN) 2021-06-23 EP claimed
WO-2020035052-A1 PYRAZINE COMPOUNDS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2020-02-20 WO claimed
EP-2621922-A1 A PROCESS FOR THE SYNTHESIS OF THIO-TRIAZOLO-GROUP CONTAINING COMPOUNDS BASF SE (DE) 2013-08-07 EP disclosed
WO-2012041858-A1 A PROCESS FOR THE SYNTHESIS OF THIO-TRIAZOLO-GROUP CONTAINING COMPOUNDS BASF SE (DE) 2012-04-05 WO disclosed