SCHEMBL9008922

SCHEMBL9008922

C=C(C)OC(=O)c1cccc(C(=O)OC(=C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.41
HSD17B10 Q99714 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
TSHR P16473 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
MAPT P10636 1/20 0.38
SLC7A5 Q01650 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17892405 0.93 CA12 (0.46) TDP1HSD17B10L3MBTL1ALDH1A1KMT2A
Isophthalic Acid SCHEMBL9008990 0.93 CA12 (0.46) TDP1HSD17B10L3MBTL1ALDH1A1KMT2A
SCHEMBL9008994 0.93 CA12 (0.46) TDP1HSD17B10L3MBTL1ALDH1A1KMT2A
SCHEMBL8925349 0.87 PARP1 (0.50) TDP1L3MBTL1ALDH1A1KMT2ARAB9A
SCHEMBL140863 0.85 TSHR (0.56) TDP1HSD17B10ATMTSHRALDH1A1
SCHEMBL123941 0.83 TDP1 (0.44) TDP1LOXL2ATML3MBTL1CYP4F2
SCHEMBL5450979 0.82 TDP1 (0.48) TDP1HSD17B10LOXL2TSHRALDH1A1
SCHEMBL10791915 0.80 KDM4E (0.41) TDP1HSD17B10ATMTSHRALDH1A1
SCHEMBL3965774 0.79 CA12 (0.61) HSD17B10L3MBTL1ALDH1A1KMT2APOLB
SCHEMBL4597257 0.78 ELANE (0.44) TDP1HSD17B10KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106624-A1 TERTIARY ALCOHOL IMIDAZOPYRAZINE BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed
WO-2016106623-A1 BENZAMIDE IMIDAZOPYRAZINE BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed
US-5534614-A Method for the preparation of amide oligomers and polybenzazole polymers therefrom THE DOW CHEMICAL COMPANY (US) 1996-07-09 US disclosed
US-5322916-A Method for the preparation of amide oligomers and polybenzazole polymers therefrom THE DOW CHEMICAL COMPANY (US) 1994-06-21 US disclosed