SCHEMBL9008944

SCHEMBL9008944

O=c1cc(-c2ccoc2)c2ccc(Sc3cc(F)cc(-c4ccc(F)cc4)c3)cc2o1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 8/20 0.68
PARP1 P09874 1/20 0.44
TPI1 P60174 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
CA12 O43570 5/20 0.35
CA9 Q16790 5/20 0.35
ALDH2 P05091 1/20 0.34
AKR1B1 P15121 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HSD17B3 P37058 1/20 0.34
SORD Q00796 1/20 0.34
PGR P06401 2/20 0.33
NOD2 Q9HC29 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9008937 0.93 ALOX5 (0.67) ALOX5PARP1TPI1PARP2CA12
SCHEMBL9008939 0.86 ALOX5 (0.67) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL9009222 0.86 ALOX5 (0.61) ALOX5PARP1TPI1PARP2CA12
SCHEMBL9008935 0.83 ALOX5 (0.51) ALOX5PARP1TPI1PARP2CA12
SCHEMBL9008946 0.81 ALOX5 (0.55) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL7803885 0.80 ALOX5 (0.77) ALOX5PARP1TPI1PARP2CA12
SCHEMBL15215912 0.79 ALOX5 (0.58) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL7812419 0.79 ALOX5 (0.76) ALOX5PARP1TPI1PARP2CA12
SCHEMBL9008978 0.76 ALOX5 (0.61) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL9008954 0.76 ALOX5 (0.59) ALOX5CA12CA9ALDH2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576338-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS AND CYTOPROTECTIVE AGENTS FOR CARDIOVASCULAR DISORDERS MERCK FROSST CANADA, INC. (CA) 1996-11-19 US claimed
US-5576338-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS AND CYTOPROTECTIVE AGENTS FOR CARDIOVASCULAR DISORDERS MERCK FROSST CANADA, INC. (CA) 1996-11-19 US disclosed