SCHEMBL9008946

SCHEMBL9008946

O=c1cc(-c2cccnc2)c2ccc(Sc3cc(F)cc(-c4ccc(F)cc4)c3)cc2o1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.55
NPC1 O15118 1/20 0.41
TNF P01375 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
NOD1 Q9Y239 1/20 0.41
CA12 O43570 5/20 0.39
CA9 Q16790 5/20 0.39
ALDH2 P05091 1/20 0.39
AKR1B1 P15121 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
HSD17B3 P37058 1/20 0.39
SORD Q00796 1/20 0.39
CYP19A1 P11511 2/20 0.38
KCNA3 P22001 1/20 0.38
TDO2 P48775 1/20 0.37
CYP17A1 P05093 1/20 0.37
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9008978 0.95 ALOX5 (0.61) ALOX5NPC1TNFPOLBRAB9A
SCHEMBL9008939 0.88 ALOX5 (0.67) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL9009222 0.87 ALOX5 (0.61) ALOX5NPC1TNFPOLBRAB9A
SCHEMBL9008944 0.81 ALOX5 (0.68) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL2994964 0.81 CA9 (0.51) NPC1TNFPOLBRAB9ANOD1
SCHEMBL9008935 0.78 ALOX5 (0.51) ALOX5CA12CA9PGR
SCHEMBL9008937 0.78 ALOX5 (0.67) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL9008954 0.77 ALOX5 (0.59) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL15215912 0.77 ALOX5 (0.58) ALOX5CA12CA9ALDH2AKR1B1
SCHEMBL2982477 0.74 KCNA3 (0.44) ALOX5NPC1TNFPOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576338-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS AND CYTOPROTECTIVE AGENTS FOR CARDIOVASCULAR DISORDERS MERCK FROSST CANADA, INC. (CA) 1996-11-19 US claimed
US-5576338-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS AND CYTOPROTECTIVE AGENTS FOR CARDIOVASCULAR DISORDERS MERCK FROSST CANADA, INC. (CA) 1996-11-19 US disclosed