SCHEMBL9008968

SCHEMBL9008968

Oc1cc(F)cc(-c2nccs2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 1/20 0.50
PDPK1 O15530 1/20 0.44
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41
HSD17B1 P14061 2/20 0.41
HSD17B2 P37059 2/20 0.41
LOXL2 Q9Y4K0 1/20 0.40
CYP2A6 P11509 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
CYP1A1 P04798 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP1B1 Q16678 2/20 0.37
SYK P43405 2/20 0.37
VCP P55072 1/20 0.37
ADRB2 P07550 1/20 0.37
ACLY P53396 1/20 0.36
CASP6 P55212 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6067979 0.87 SMPD3 (0.58) SMPD3PDPK1LOXL2CYP2A6ESR1
SCHEMBL753260 0.73 PDPK1 (0.60) SMPD3PDPK1HSD17B1HSD17B2LOXL2
SCHEMBL31609722 0.73 PDPK1 (0.60) SMPD3PDPK1HSD17B1HSD17B2LOXL2
SCHEMBL173979 0.73 PDPK1 (0.60) PDPK1LOXL2CYP2A6CYP1A1CYP1A2
SCHEMBL252833 0.73 CYP2A6 (0.53) SMPD3PDPK1LOXL2CYP2A6CYP1A1
SCHEMBL15668605 0.71 CYP1A1 (0.47) SMPD3PDPK1CYP1A1CYP1A2CYP1B1
SCHEMBL4589649 0.71 PDPK1 (0.63) SMPD3PDPK1LOXL2CYP2A6CYP1A1
SCHEMBL466426 0.71 PDPK1 (0.63) SMPD3PDPK1LOXL2CYP2A6ESR1
Ammonia Solution, Strong SCHEMBL29239355 0.69 PDPK1 (0.61) SMPD3PDPK1LOXL2CYP2A6ESR1
SCHEMBL15668645 0.69 CYP1A1 (0.44) SMPD3PDPK1CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120328691-A1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME LLC 2012-12-27 US disclosed
US-5576338-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS AND CYTOPROTECTIVE AGENTS FOR CARDIOVASCULAR DISORDERS MERCK FROSST CANADA, INC. (CA) 1996-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120328691-A1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MAPK15, CDK15, MAPKAPK5 SMPD3 3384/4885PDPK1 193/4885CA12 3583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.