SCHEMBL9010372

SCHEMBL9010372

C=CCN1C(=O)c2cccnc2Nc2ncccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
BRD4 O60885 1/20 0.47
CASP3 P42574 1/20 0.46
LMNA P02545 2/20 0.45
PKM P14618 2/20 0.45
MAPT P10636 1/20 0.45
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CYP1A2 P05177 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KMT2A Q03164 3/20 0.39
GALR3 O60755 1/20 0.39
CHEK1 O14757 1/20 0.38
MEN1 O00255 2/20 0.38
MAPK1 P28482 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301745 0.82 ALDH1A1 (0.54) ALDH1A1BRD4LMNAPKMMAPT
SCHEMBL8304689 0.75 ALDH1A1 (0.52) ALDH1A1BRD4CASP3MAPTGAA
SCHEMBL9101209 0.73 TP53 (0.54) ALDH1A1BRD4CASP3LMNAPKM
SCHEMBL9369241 0.73 BRD4 (0.50) ALDH1A1BRD4CASP3LMNAPKM
SCHEMBL8790523 0.70 ALDH1A1 (0.79) ALDH1A1CYP1A2SMN1; SMN2
SCHEMBL8790081 0.70 ALDH1A1 (0.71) ALDH1A1BRD4MAPTKDM4EGAA
SCHEMBL9431569 0.70 ALDH1A1 (0.57) ALDH1A1CYP1A2SMN1; SMN2
SCHEMBL17667422 0.70 CASP3 (0.59) ALDH1A1BRD4CASP3LMNAPKM
SCHEMBL8936638 0.69 BRD4 (0.44) ALDH1A1BRD4CASP3LMNAPKM
SCHEMBL170913 0.69 CASP3 (0.85) ALDH1A1CASP3LMNAPKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532358-A Method for preparing alkyl-5,11-dihydro-6h-dipyrido[3,2-B:2',3'-E] [1,4] diazepin-6-ones BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1996-07-02 US disclosed