SCHEMBL9011190

SCHEMBL9011190

O=C(O)CCCc1cccc(C2CCN(C(=O)c3cccc4ccccc34)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.52
TPSAB1 Q15661 10/20 0.52
AVPR1A P37288 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9011116 0.95 CCR5 (0.53) CCR5TPSAB1AVPR1AMEN1KMT2A
SCHEMBL9011078 0.89 CCR5 (0.54) CCR5AVPR1ACYP1A2CYP2D6CYP2C19
SCHEMBL9011020 0.88 CCR5 (0.55) CCR5TPSAB1AVPR1AMEN1KMT2A
SCHEMBL9011270 0.84 DRD4 (0.59) CYP1A2
SCHEMBL9011180 0.84 CCR5 (0.55) CCR5AVPR1ACYP2D6MEN1KMT2A
SCHEMBL7813354 0.84 CCR5 (0.51) CCR5TPSAB1AVPR1AMEN1KMT2A
SCHEMBL27295602 0.83 CCR5 (0.66) CCR5AVPR1AMEN1KMT2AKDM4E
SCHEMBL7817613 0.82 CCR5 (0.51) CCR5TPSAB1AVPR1AMEN1KMT2A
SCHEMBL9011219 0.81 ALDH1A1 (0.50) CCR5AVPR1AMEN1KMT2AKDM4E
SCHEMBL9011047 0.81 ALDH1A1 (0.55) AVPR1ACYP1A2CYP2D6CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532371-A SIDE EFFECT REDUCTION SS PHARMACEUTICAL CO., LTD. (JP) 1996-07-02 US disclosed
US-5411972-A Arylamide derivatives for treating hyperlipemia SS PHARMACEUTICAL CO., LTD. (JP) 1995-05-02 US disclosed
EP-0607536-A1 Arylamide derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1994-07-27 EP disclosed