SCHEMBL9011180

SCHEMBL9011180

O=C(O)CCc1ccc(C2CCN(C(=O)c3cccc4ccccc34)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.55
CYP2D6 P10635 1/20 0.52
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
HIF1A Q16665 1/20 0.51
CHRM2 P08172 3/20 0.50
AVPR1A P37288 1/20 0.50
HRH1 P35367 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
S1PR1 P21453 1/20 0.46
CCR3 P51677 1/20 0.45
DRD4 P21917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9011078 0.94 CCR5 (0.54) CCR5CYP2D6ALDH1A1KDM4EMEN1
SCHEMBL9011116 0.89 CCR5 (0.53) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9010977 0.89 CCR5 (0.57) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL27295602 0.86 CCR5 (0.66) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9011190 0.84 CCR5 (0.52) CCR5CYP2D6ALDH1A1KDM4EMEN1
SCHEMBL7814084 0.84 HRH1 (0.56) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL7809741 0.84 HRH1 (0.56) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9010990 0.82 ALDH1A1 (0.51) CCR5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9011199 0.82 ALDH1A1 (0.58) ALDH1A1KDM4EMEN1KMT2AHIF1A
SCHEMBL7817573 0.81 ALDH1A1 (0.59) CCR5CYP2D6ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1035178-C Arylamide derivatives SS PHARMACEUTICAL CO (JP) 1997-06-18 CN disclosed
US-5532371-A SIDE EFFECT REDUCTION SS PHARMACEUTICAL CO., LTD. (JP) 1996-07-02 US disclosed
US-5411972-A Arylamide derivatives for treating hyperlipemia SS PHARMACEUTICAL CO., LTD. (JP) 1995-05-02 US disclosed
EP-0607536-A1 Arylamide derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1994-07-27 EP disclosed