SCHEMBL9011479

SCHEMBL9011479

CCC(C#N)(CC(N)=O)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.33
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 2/20 0.31
CYP1A2 P05177 2/20 0.31
KMT2A Q03164 2/20 0.31
TSHR P16473 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836697 0.83 TSHR (0.39) ALDH1A1MEN1CYP1A2KMT2ATSHR
SCHEMBL1341696 0.83 ALDH1A1 (0.37) MCL1ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL3108109 0.76 ALDH1A1 (0.35) MCL1ALDH1A1TSHR
SCHEMBL2147379 0.75 ALDH1A1 (0.32) MCL1ALDH1A1TSHR
SCHEMBL3542104 0.75 ALDH1A1 (0.32) MCL1ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL8164857 0.72 GRM2 (0.32) ALDH1A1TSHR
SCHEMBL17499002 0.71
Water SCHEMBL31084442 0.70 MCL1 (0.34) MCL1ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL4734754 0.70 MCL1 (0.34) MCL1ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL10882205 0.69 MEN1 (0.30) ALDH1A1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421946-B1 3-indolepyruvic acid derivatives their method of production and therapeutic use POLIFARMA SPA (IT) 1996-11-20 EP disclosed
EP-0421946-A2 3-indolepyruvic acid derivatives their method of production and therapeutic use POLIFARMA S.p.A. (IT) 1991-04-10 EP disclosed