SCHEMBL9012744

SCHEMBL9012744

COc1ccc(-c2[c]cccc2S(C)(=O)=O)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ABCB11 O95342 1/20 0.38
NR1H3 Q13133 1/20 0.37
AR P10275 2/20 0.36
S1PR1 P21453 1/20 0.35
ERAP1 Q9NZ08 1/20 0.35
PGR P06401 1/20 0.35
CTSS P25774 3/20 0.35
CTSK P43235 3/20 0.35
AXL P30530 1/20 0.34
KIF11 P52732 1/20 0.34
PTGS2 P35354 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9119744 0.84 PTGS2 (0.44) SMN1; SMN2LMNAHPGDHTTNPSR1
SCHEMBL9012907 0.84 PTGS2 (0.50) SMN1; SMN2PTGS2PTGS1
SCHEMBL9012633 0.82 NOTUM (0.40) NR1H2LMNAHTTNPSR1KMT2A
SCHEMBL9012728 0.82 PTGS2 (0.46) NR1H2SMN1; SMN2LMNAHTTNPSR1
SCHEMBL6402326 0.81 PTGS2 (0.52) SMN1; SMN2KMT2APTGS2PTGS1
SCHEMBL9012755 0.81 PTGS2 (0.44) SMN1; SMN2LMNAHPGDTP53PTGS2
SCHEMBL9012598 0.76 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL9013542 0.76 PTGS2 (0.40) NR1H2SMN1; SMN2LMNANPSR1KMT2A
SCHEMBL9013714 0.75 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL9117190 0.74 PTGS2 (0.41) SMN1; SMN2TP53PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743938-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-27 EP disclosed
WO-1995021817-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-08-17 WO disclosed