SCHEMBL9013438

SCHEMBL9013438

CC(=O)OCc1cc(Br)ncc1Br

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
CYP3A4 P08684 1/20 0.36
CA2 P00918 2/20 0.36
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 2/20 0.35
PKM P14618 2/20 0.33
MAPT P10636 4/20 0.32
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
NOTUM Q6P988 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28847143 0.83 NQO1 (0.36) KDM4E
SCHEMBL19683552 0.75 ALDH1A1 (0.44) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL21358386 0.74 NOS3 (0.36)
SCHEMBL28049660 0.72 ALDH1A1 (0.43) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL20568246 0.72 ALDH1A1 (0.43) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL1315960 0.72 HSD17B10 (0.41) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL3293016 0.71 ALDH1A1 (0.52) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL5936414 0.71 CYP3A4 (0.55) ALDH1A1CYP3A4CA2KDM4EHSD17B10
SCHEMBL22899909 0.71
SCHEMBL1315783 0.71 NOTUM (0.40) ALDH1A1CYP3A4CA2KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536745-A (Hetero)-aryl ketones derivatives with antibacterial properties SMITHKLINE BEECHAM P.L.C. (GB) 1996-07-16 US disclosed
EP-0652875-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1995-05-17 EP disclosed
WO-1994002478-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1994-02-03 WO disclosed