SCHEMBL9013541

SCHEMBL9013541

COc1ccc(-c2nc(C)cc(O)n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.54
NPC1 O15118 7/20 0.50
RAB9A P51151 5/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
KDM4E B2RXH2 4/20 0.50
TP53 P04637 3/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 1/20 0.50
DYRK1A Q13627 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
ATM Q13315 1/20 0.47
MAPT P10636 5/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MAPK1 P28482 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2118153 0.89 ESR2 (0.52) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL17720570 0.87 KDM4E (0.57) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL10968094 0.82 NPC1 (0.46) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL632828 0.79 LMNA (0.64) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL9013358 0.79 DYRK1A (0.54) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL9013519 0.79 KDM4E (0.55) SMN1; SMN2KDM4ETP53ALDH1A1HPGD
SCHEMBL9013731 0.79 NPC1 (0.47) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL2577307 0.78 LMNA (0.61) ABCG2NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL11515085 0.78 ABCG2 (0.48) ABCG2NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL9013267 0.77 ABCG2 (0.62) ABCG2NPC1RAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589477-A LEARNING ENHANCEMENT, CNS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-12-31 US disclosed
EP-0555478-A1 PYRIMIDINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-18 EP disclosed
EP-0153746-B1 3-AMINO-2-HYDROXYPROPYL DERIVATIVES OF PYRIMIDIN-4-ONE MERCK & CO. INC. (US) 1990-11-22 EP disclosed
US-4598149-A ADRENERGIC BLOCKING AGENTS MERCK & CO., INC. (US) 1986-07-01 US disclosed
EP-0153746-A2 3-Amino-2-hydroxypropyl derivatives of pyrimidin-4-one MERCK & CO. INC. (US) 1985-09-04 EP disclosed