SCHEMBL9014334

SCHEMBL9014334

COc1ccc2c(c1)C(CC(=O)N1CCC(c3ccc(OC)c(OC)c3)CC1)CO2

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.46
PDE4B Q07343 11/20 0.45
CYP3A4 P08684 2/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
QDPR P09417 1/20 0.43
PDE4A P27815 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
LMNA P02545 1/20 0.41
ADAM17 P78536 1/20 0.41
ADAMTS5 Q9UNA0 1/20 0.41
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014309 0.89 KCNH2 (0.59) KCNH2PDE4BQDPR
SCHEMBL9014392 0.82 KCNH2 (0.65) KCNH2CYP3A4MEN1MAPTKMT2A
SCHEMBL9014717 0.79 ABCB1 (0.48) PDE4BMEN1KMT2AQDPR
SCHEMBL9014397 0.79 PDE4B (0.44) PDE4BQDPRPDE4APDE4CPDE4D
SCHEMBL9014711 0.75 PTGDR2 (0.51) KCNH2PDE4BQDPRPDE4APDE4C
SCHEMBL9628106 0.74 PPARD (0.56)
SCHEMBL9014779 0.74 KCNH2 (0.70) KCNH2
SCHEMBL9014710 0.73 PTGDR2 (0.52) PDE4BKMT2ASMN1; SMN2QDPR
SCHEMBL9014339 0.72 PDE4B (0.46) KCNH2PDE4BQDPRPDE4APDE4C
SCHEMBL9014422 0.71 FFAR1 (0.48) KCNH2MAPTSMN1; SMN2LMNAADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed