SCHEMBL9014384

SCHEMBL9014384

COc1ccc(C2CCN(C(=O)CC3CCNc4ccc(Cl)cc43)CC2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 8/20 0.47
ADAMTS5 Q9UNA0 3/20 0.45
PDE4B Q07343 8/20 0.44
CCR2 P41597 1/20 0.43
QDPR P09417 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014339 0.88 PDE4B (0.46) ADAM17ADAMTS5PDE4BQDPRLMNA
SCHEMBL9014397 0.84 PDE4B (0.44) ADAM17ADAMTS5PDE4BQDPRLMNA
SCHEMBL9233397 0.83 ADAM17 (0.47) ADAM17ADAMTS5PDE4BQDPRLMNA
SCHEMBL9014784 0.82 KCNH2 (0.55) CCR2QDPR
SCHEMBL9014711 0.75 PTGDR2 (0.51) ADAM17ADAMTS5PDE4BQDPR
SCHEMBL9014710 0.74 PTGDR2 (0.52) PDE4BQDPR
SCHEMBL9014717 0.72 ABCB1 (0.48) PDE4BQDPR
SCHEMBL9014309 0.72 KCNH2 (0.59) PDE4BQDPR
SCHEMBL9014334 0.70 KCNH2 (0.46) ADAM17ADAMTS5PDE4BQDPRLMNA
SCHEMBL22062947 0.70 ADAM17 (0.62) ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed