Choline

Choline

SCHEMBL9015240

C[N+](C)(C)CCO.C[N+](C)(C)CCO.[O-]B([O-])OCCCC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of Choline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.38
CHRM4 P08173 4/20 0.38
CHRM1 P11229 4/20 0.38
CHRM3 P20309 4/20 0.38
CHRM5 P08912 2/20 0.38
KIF11 P52732 10/20 0.37
KCNH2 Q12809 2/20 0.36
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SCN1A P35498 3/20 0.32
SCN2A Q99250 3/20 0.32
SCN3A Q9NY46 3/20 0.32
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Choline SCHEMBL9015244 0.88 CHRM2 (0.38) CHRM2CHRM4CHRM1CHRM3CHRM5
Tetramethylammonium Ion SCHEMBL2428731 0.87 KIF11 (0.44) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL9685834 0.86 KIF11 (0.36) CHRM2CHRM4CHRM1CHRM3CHRM5
Lithium Ion SCHEMBL3623447 0.83 KIF11 (0.48) KIF11KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL9686702 0.83 KDM4E (0.45) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL1092325 0.81 SCN1A (0.41) CHRM2CHRM4CHRM1CHRM3CHRM5
Tetrylammonium SCHEMBL3297055 0.81 KIF11 (0.41) CHRM2CHRM4CHRM1CHRM3CHRM5
Tetrabuthylammonium SCHEMBL125284 0.80 KIF11 (0.38) CHRM2CHRM4CHRM1CHRM3CHRM5
Choline SCHEMBL9015229 0.77 KIF11 (0.43) CHRM2CHRM4CHRM1CHRM3CHRM5
Tetramethylammonium Ion SCHEMBL1146377 0.76 KIF11 (0.44) CHRM2CHRM4CHRM1CHRM3CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0572524-B1 RED SENSITIVE PHOTOPOLYMERIZABLE COMPOSITIONS DU PONT (US) 1996-12-18 EP disclosed
EP-0569488-A1 BORATE COINITIATORS FOR PHOTOPOLYMERIZABLE COMPOSITIONS. DU PONT (US) 1993-11-18 EP disclosed
US-5147758-A Containing squarylium dye, boron anion initiator E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-09-15 US disclosed
WO-1992013900-A1 BORATE COINITIATORS FOR PHOTOPOLYMERIZABLE COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-08-20 WO disclosed