SCHEMBL9016301

SCHEMBL9016301

CCc1cc(CCNC(=O)Oc2ccccc2)c(OC)nc1C

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.52
NPC1 O15118 1/20 0.52
GAA P10253 1/20 0.52
RAB9A P51151 1/20 0.52
FAAH O00519 5/20 0.52
TRPV1 Q8NER1 1/20 0.47
BRD4 O60885 2/20 0.43
MTNR1A P48039 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058202 0.94 FAAH (0.47) TAAR1NPC1GAARAB9AFAAH
SCHEMBL9016298 0.92 BRD4 (0.47) TAAR1NPC1GAARAB9AFAAH
SCHEMBL8701292 0.89 ALDH1A1 (0.43) TAAR1NPC1GAARAB9AFAAH
SCHEMBL6953240 0.81 KMT2A (0.46) NPC1GAARAB9ATRPV1
SCHEMBL9058102 0.80 FAAH (0.43) FAAHBRD4
SCHEMBL8699410 0.79 MAPT (0.40) NPC1GAARAB9A
SCHEMBL6966654 0.76 ALDH1A1 (0.43) NPC1GAARAB9AFAAHTRPV1
SCHEMBL8699180 0.76 HPGD (0.41) GAA
SCHEMBL8699066 0.74 RAB9A (0.44) NPC1GAARAB9AFAAHTRPV1
SCHEMBL8703454 0.74 MAPK1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749425-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARM. CO., LTD. (KR) 1996-12-27 EP disclosed
WO-1996021648-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1996-07-18 WO disclosed