SCHEMBL10189200

SCHEMBL10189200

COC(=O)CC1CCC(c2ccc(-c3ccc(-c4nc5ccc(Cl)cc5[nH]4)nc3)cc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 0.71
SOAT1 P35610 6/20 0.66
KCNH2 Q12809 13/20 0.57
ADORA2A P29274 1/20 0.50
CYP2C8 P10632 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189566 0.83 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902557 0.83 DGAT1 (0.86) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902206 0.80 DGAT1 (0.61) DGAT1SOAT1KCNH2
SCHEMBL902450 0.79 DGAT1 (0.60) DGAT1SOAT1
SCHEMBL901744 0.79 DGAT1 (0.58) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901747 0.79 DGAT1 (0.70) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL4312086 0.77 DGAT1 (0.47) DGAT1SOAT1
SCHEMBL901177 0.77 DGAT1 (0.56) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189107 0.76 DGAT1 (0.86) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL181024 0.76 DGAT1 (0.48) DGAT1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed