SCHEMBL9017539

SCHEMBL9017539

Cc1c(S(C)(=O)=O)[nH]c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.59
CNR1 P21554 9/20 0.54
DAO P14920 1/20 0.49
DDO Q99489 1/20 0.49
PTGS2 P35354 3/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
RAB9A P51151 1/20 0.44
GAA P10253 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GPR3 P46089 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 1/20 0.42
HPGD P15428 1/20 0.42
GFER P55789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4238498 0.83 CNR1 (0.52) AHRCNR1DAODDOPTGS2
SCHEMBL28833067 0.81 AHR (0.59) AHRCNR1DAODDOCYP1A2
SCHEMBL8780773 0.80 CNR1 (0.51) AHRCNR1DAODDOPTGS2
SCHEMBL9017534 0.79 PTGS2 (0.43) AHRCNR1PTGS2CYP1A2CYP2C19
SCHEMBL8307123 0.78 PTGS2 (0.45) AHRCNR1PTGS2CYP1A2CYP2C19
SCHEMBL154593 0.74 AHR (1.00) AHRDAODDOCYP1A2CYP2C19
SCHEMBL29420757 0.74 AHR (1.00) AHRDAODDOCYP1A2CYP2C19
SCHEMBL6202865 0.74 AHR (0.55) AHRPTGS2CYP1A2CYP2C19TNKS2
SCHEMBL8610115 0.74 PTGS2 (0.69) AHRPTGS2
SCHEMBL7195762 0.72 AHR (0.70) AHRDAODDOCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed