SCHEMBL9017534

SCHEMBL9017534

[CH2]c1c(S(C)(=O)=O)[nH]c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.43
AHR P35869 1/20 0.42
ALDH1A1 P00352 3/20 0.41
GPR3 P46089 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 2/20 0.41
GLA P06280 1/20 0.41
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CNR1 P21554 2/20 0.39
CYP1A2 P05177 3/20 0.39
TNKS2 Q9H2K2 2/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 1/20 0.38
TNKS O95271 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307123 0.80 PTGS2 (0.45) PTGS2AHRALDH1A1GPR3HSD17B10
SCHEMBL9017539 0.79 AHR (0.59) PTGS2AHRALDH1A1GPR3HSD17B10
SCHEMBL5781155 0.74 AHR (0.61) AHRALDH1A1GPR3HSD17B10KDM4E
SCHEMBL8089249 0.70 ALDH1A1 (0.50) AHRALDH1A1GPR3HSD17B10KDM4E
SCHEMBL9260741 0.69 ALDH1A1 (0.40) PTGS2ALDH1A1KDM4EGAAHPGD
SCHEMBL6202865 0.69 AHR (0.55) PTGS2AHRALDH1A1GPR3HSD17B10
SCHEMBL4238498 0.67 CNR1 (0.52) PTGS2AHRALDH1A1GPR3HSD17B10
SCHEMBL8084325 0.66 ALDH1A1 (0.50) AHRALDH1A1GPR3HSD17B10KDM4E
SCHEMBL7495853 0.66 ALDH1A1 (0.50) AHRALDH1A1GPR3HSD17B10KDM4E
SCHEMBL8083535 0.66 ALDH1A1 (0.50) AHRALDH1A1GPR3HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed