SCHEMBL9017869

SCHEMBL9017869

CN(C)C(=O)Oc1cnccc1N=CN1CCSCC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 5/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RAB9A P51151 2/20 0.33
PKM P14618 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
BCHE P06276 1/20 0.32
MAOA P21397 1/20 0.32
ACHE P22303 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9017868 1.00 NCEH1 (0.33) NCEH1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9017864 0.92 BCHE (0.38) NCEH1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9017860 0.92 BCHE (0.38) NCEH1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9017892 0.91 ACHE (0.39) NCEH1RAB9APKMNPC1TSHR
SCHEMBL9017889 0.91 ACHE (0.39) NCEH1RAB9APKMNPC1TSHR
SCHEMBL9017875 0.91 ACHE (0.39) NCEH1RAB9APKMNPC1TSHR
SCHEMBL9017879 0.91 ACHE (0.39) NCEH1RAB9APKMNPC1TSHR
SCHEMBL9017878 0.87 GAA (0.37) NCEH1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9017874 0.87 GAA (0.37) NCEH1KDM4EALDH1A1HPGDHSD17B10
Dimethylcarbate SCHEMBL9680307 0.80 KDM4E (0.30) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477903-B1 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-04-03 EP disclosed
EP-0477903-A2 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-04-01 EP disclosed