SCHEMBL901856

SCHEMBL901856

Nc1ncccc1-c1cc(C(F)(F)F)ccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.51
NOS2 P35228 1/20 0.51
MAP4K4 O95819 1/20 0.42
TLR7 Q9NYK1 2/20 0.40
RIPK1 Q13546 1/20 0.39
GRM5 P41594 1/20 0.39
TOP1 P11387 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
GSK3B P49841 1/20 0.37
DYRK1A Q13627 1/20 0.37
MAT2A P31153 1/20 0.37
KIF11 P52732 1/20 0.37
CBFB Q13951 1/20 0.37
SLC40A1 Q9NP59 2/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
TGFBR1 P36897 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17895180 0.78 TLR7 (0.46) NOS3NOS2TLR7
SCHEMBL3140455 0.77 MAP4K4 (0.63) NOS3NOS2MAP4K4TLR7RIPK1
SCHEMBL28726696 0.77 NPC1 (0.49) NOS3NOS2MAP4K4MAPK1DYRK1A
SCHEMBL810884 0.76 NOS3 (0.61) NOS3NOS2GRM5TSHRMAPK1
SCHEMBL322548 0.75 HSD17B10 (0.50) NOS3NOS2TLR7TSHRMAPK1
SCHEMBL972297 0.75 HSD11B1 (0.45) NOS3NOS2MAPK1GSK3BMAT2A
SCHEMBL29888283 0.75 MKNK1 (0.54) MAP4K4TLR7RIPK1TOP1KIF11
SCHEMBL7089225 0.74 NOS3 (0.51) NOS3NOS2TSHRMAPK1GSK3B
SCHEMBL24363083 0.74 KDM4E (0.54) NOS3NOS2TLR7GRM5MAPK1
SCHEMBL5685446 0.73 NOS3 (0.50) NOS3NOS2TSHRMAPK1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900665-A1 TRIAZOLYL DERIVATIVES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-08-05 EP disclosed