SCHEMBL9020070

SCHEMBL9020070

O=C(OCc1ccc([N+](=O)[O-])cc1)N1CCC([C@@H]2C[C@@H](O)CN2C(=O)OCc2ccc([N+](=O)[O-])cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.43
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
RAB9A P51151 2/20 0.39
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
NPC1 O15118 1/20 0.38
ATM Q13315 1/20 0.38
OPRK1 P41145 1/20 0.38
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020352 0.95 CCR5 (0.42) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL9020217 0.90 CCR5 (0.43) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL9399937 0.88 CCR5 (0.45) CCR5ALDH1A1MAPTHPGDTDP1
SCHEMBL9020408 0.86 CCR5 (0.44) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL9020729 0.85 CCR5 (0.42) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL9020800 0.85 CCR5 (0.42) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL5723982 0.83 ALDH1A1 (0.47) ALDH1A1MAPTHPGDLMNATDP1
SCHEMBL5723978 0.83 ALDH1A1 (0.47) ALDH1A1MAPTHPGDLMNATDP1
SCHEMBL4476414 0.83 ALDH1A1 (0.47) ALDH1A1MAPTHPGDLMNATDP1
SCHEMBL9399827 0.81 ALDH1A1 (0.45) CCR5ALDH1A1MAPTHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449191-B1 2-(Substituted pyrrolidinylthio)carbapenem derivatives BANYU PHARMA CO LTD (JP) 1996-07-03 EP disclosed
US-5438054-A Antibacterial agent BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-01 US disclosed
US-5374720-A A thienamycins bactericides has nontoxic, side effect reduction against the kidney and central nervous system BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-12-20 US disclosed
WO-1991014687-A1 2-(SUBSTITUTED PYRROLIDINYLTHIO)CARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-10-03 WO disclosed
EP-0449191-A1 2-(Substituted pyrrolidinylthio)carbapenem derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-10-02 EP disclosed