SCHEMBL9020729

SCHEMBL9020729

CC(=O)S[C@H]1C[C@@H](C2CCN(C(=O)OCc3ccc([N+](=O)[O-])cc3)C2)N(C(=O)OCc2ccc([N+](=O)[O-])cc2)C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.42
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ATM Q13315 1/20 0.37
KCNJ1 P48048 1/20 0.37
KCNH2 Q12809 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
HTT P42858 1/20 0.36
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020004 0.95 CCR5 (0.41) CCR5ALDH1A1MAPTHPGDKDM4E
SCHEMBL9020939 0.94 CCR5 (0.44) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL9399680 0.90 CCR5 (0.42) CCR5ALDH1A1MAPTHPGDATM
SCHEMBL9020070 0.85 CCR5 (0.43) CCR5ALDH1A1MAPTHPGDKDM4E
SCHEMBL9020217 0.85 CCR5 (0.43) CCR5ALDH1A1MAPTHPGDKDM4E
SCHEMBL195525 0.85 ALDH1A1 (0.44) ALDH1A1MAPTHPGDKDM4ELMNA
SCHEMBL9519199 0.83 PREP (0.43) CCR5ALDH1A1MAPTHPGDATM
SCHEMBL9020078 0.83 RAB9A (0.38) CCR5ALDH1A1MAPTHPGDLMNA
SCHEMBL7799332 0.83 ALDH1A1 (0.37) ALDH1A1MAPTHPGDKDM4ELMNA
SCHEMBL9519307 0.83 PREP (0.42) CCR5ALDH1A1MAPTHPGDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449191-B1 2-(Substituted pyrrolidinylthio)carbapenem derivatives BANYU PHARMA CO LTD (JP) 1996-07-03 EP disclosed
US-5438054-A Antibacterial agent BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-01 US disclosed
US-5374720-A A thienamycins bactericides has nontoxic, side effect reduction against the kidney and central nervous system BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-12-20 US disclosed
WO-1991014687-A1 2-(SUBSTITUTED PYRROLIDINYLTHIO)CARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-10-03 WO disclosed
EP-0449191-A1 2-(Substituted pyrrolidinylthio)carbapenem derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-10-02 EP disclosed