SCHEMBL9020179

SCHEMBL9020179

CN1C(=O)CC([C@@H]2C[C@@H](O[Si](C)(C)C(C)(C)C)CN2C(=O)OCc2ccc([N+](=O)[O-])cc2)C1=O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CCR5 P51681 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PAX8 Q06710 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020242 0.88 ALDH1A1 (0.43) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL9020149 0.84 ATM (0.44) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL9020561 0.83 ALDH1A1 (0.42) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL9020154 0.82 ALDH1A1 (0.41) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL9399096 0.82 ALDH1A1 (0.43) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL9020556 0.81 CCR5 (0.43) ALDH1A1MAPTHPGDCCR5NPC1
SCHEMBL9399315 0.80 ALDH1A1 (0.42) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL5233422 0.80 ALDH1A1 (0.40) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL8923324 0.80 ALDH1A1 (0.40) ALDH1A1MAPTHPGDATMTDP1
SCHEMBL9366344 0.80 ALDH1A1 (0.40) ALDH1A1MAPTHPGDATMTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449191-B1 2-(Substituted pyrrolidinylthio)carbapenem derivatives BANYU PHARMA CO LTD (JP) 1996-07-03 EP disclosed
US-5438054-A Antibacterial agent BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-01 US disclosed
US-5374720-A A thienamycins bactericides has nontoxic, side effect reduction against the kidney and central nervous system BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-12-20 US disclosed
WO-1991014687-A1 2-(SUBSTITUTED PYRROLIDINYLTHIO)CARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-10-03 WO disclosed
EP-0449191-A1 2-(Substituted pyrrolidinylthio)carbapenem derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-10-02 EP disclosed