SCHEMBL9020786

SCHEMBL9020786

Cc1cccc2c1C(B(O)O)c1ccccc1-2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
HTR7 P34969 1/20 0.35
HTR2B P41595 1/20 0.35
GPR3 P46089 1/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
ATM Q13315 1/20 0.34
POLB P06746 1/20 0.33
KDM4E B2RXH2 2/20 0.33
PBRM1 Q86U86 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MYC P01106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18343745 0.83 GPR3 (0.32) GPR3KMT2AMEN1POLBLMNA
SCHEMBL5034116 0.82 GPR3 (0.34) GPR3KMT2APOLB
SCHEMBL1044055 0.78 GPR3 (0.41) ALDH1A1GPR3KMT2AMEN1POLB
SCHEMBL29953549 0.78 GPR3 (0.41) ALDH1A1GPR3KMT2AMEN1POLB
SCHEMBL11783880 0.77 HTR2B (0.51) ALDH1A1HTR7HTR2BGPR3KMT2A
SCHEMBL9020869 0.76 PDCD1 (0.39)
Water SCHEMBL27413384 0.76 HTR2B (0.50) ALDH1A1HTR7HTR2BGPR3KMT2A
Methyl Alcohol SCHEMBL14815699 0.74 ALDH1A1 (0.38) ALDH1A1HTR7HTR2BGPR3KMT2A
SCHEMBL447441 0.73 MEN1 (0.35) ALDH1A1KMT2AMEN1POLBMAPT
SCHEMBL358532 0.73 GPR3 (0.39) ALDH1A1HTR7HTR2BGPR3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0669921-A4 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION. MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0669921-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO. INC. (US) 1995-09-06 EP disclosed
US-5442057-A Preparation of 2-aryl carbapenems via a boronic acid coupling reaction DECAMP ANN (US) 1995-08-15 US disclosed
US-5338875-A Boron containing intermediates useful in the preparation of carbapenems MERCK & CO., INC. (US) 1994-08-16 US disclosed
WO-1994011372-A1 PREPARATION OF 2-ARYL CARBAPENEMS VIA A BORONIC ACID COUPLING REACTION MERCK & CO., INC. (US) 1994-05-26 WO disclosed