SCHEMBL9020901

SCHEMBL9020901

CC(=O)Nc1nc(Cl)c2c(ncn2COC(COCc2ccccc2)COC(=O)C(C)(C)C)n1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.48
ACHE P22303 3/20 0.41
NPR3 P17342 2/20 0.39
ADORA3 P0DMS8 7/20 0.35
ADORA2A P29274 7/20 0.35
ADORA1 P30542 7/20 0.35
PRKCA P17252 1/20 0.35
PRKCD Q05655 1/20 0.35
TBXAS1 P24557 1/20 0.32
HPGD P15428 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021602 0.90 ACHE (0.40) BCHEACHENPR3ADORA3ADORA2A
SCHEMBL9021161 0.89 BCHE (0.50) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9019704 0.86 NPR3 (0.40) BCHENPR3PRKCAPRKCDTBXAS1
SCHEMBL9575361 0.82 BCHE (0.48) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9021427 0.80 ACHE (0.42) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9021416 0.80 ACHE (0.41) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9021782 0.78 ACHE (0.43) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9021299 0.78 ACHE (0.42) BCHEACHEADORA3ADORA2AADORA1
SCHEMBL9021599 0.77 ACHE (0.41) BCHEACHE
SCHEMBL10364108 0.76 ACHE (0.40) ACHENPR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452680-B1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AG (DE) 1996-11-06 EP disclosed
EP-0452680-A1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-23 EP disclosed