SCHEMBL902148

SCHEMBL902148

CCC(CCC(C)CC(=O)NC)c1ccc(C2=CC=C(c3nc4cc(C(F)(F)F)ccc4[nH]3)CC2)cc1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 2/20 0.33
NPBWR1 P48145 4/20 0.32
DGAT1 O75907 3/20 0.32
SOAT1 P35610 1/20 0.32
KCNH2 Q12809 3/20 0.32
PDE2A O00408 3/20 0.32
CHEK2 O96017 1/20 0.31
MMP1 P03956 1/20 0.31
MMP3 P08254 1/20 0.31
MMP7 P09237 1/20 0.31
ACACB O00763 1/20 0.31
ACACA Q13085 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902608 0.71 DGAT1 (0.45) NPBWR1DGAT1SOAT1KCNH2PDE2A
SCHEMBL10381238 0.66 NPBWR1 (0.42) NPBWR1DGAT1SOAT1KCNH2
SCHEMBL15245153 0.66 DGAT1 (0.54) NPBWR1DGAT1SOAT1KCNH2CHEK2
SCHEMBL20661007 0.65 PARP1 (0.53) NPBWR1DGAT1KCNH2
SCHEMBL20661102 0.62 KDM4E (0.59) NPBWR1DGAT1KCNH2
SCHEMBL20660944 0.61 EGFR (0.58) NPBWR1DGAT1KCNH2
SCHEMBL10576428 0.61 PKN1 (0.46) CHEK2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL15245155 0.61 DGAT1 (0.56) NPBWR1DGAT1SOAT1KCNH2CHEK2
SCHEMBL15245140 0.61 DGAT1 (0.67) NPBWR1DGAT1SOAT1KCNH2
SCHEMBL21263976 0.60 NOTUM (0.52) NPBWR1DGAT1SOAT1KCNH2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed