SCHEMBL902608

SCHEMBL902608

CNC(=O)CC1CCC(C2=CC=C(C3=CC=C(c4nc5cc(C(F)(F)F)ccc5[nH]4)CC3)CC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 12/20 0.45
SOAT1 P35610 3/20 0.45
KCNH2 Q12809 5/20 0.37
ADORA2A P29274 1/20 0.36
CSNK1D P48730 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CYP2C9 P11712 3/20 0.35
CYP3A4 P08684 2/20 0.35
IDO1 P14902 1/20 0.35
FFAR4 Q5NUL3 2/20 0.32
PDE2A O00408 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPBWR1 P48145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10188922 0.76 DGAT1 (0.41) DGAT1SOAT1KCNH2ADORA2AFFAR4
SCHEMBL902786 0.75 DGAT1 (0.40) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902149 0.72 DGAT1 (0.62) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL902559 0.72 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL901617 0.71 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902148 0.71 SOS1 (0.33) DGAT1SOAT1KCNH2CYP2C9CYP3A4
SCHEMBL902020 0.70 DGAT1 (0.59) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL10381238 0.69 NPBWR1 (0.42) DGAT1SOAT1KCNH2NPBWR1
SCHEMBL10189190 0.69 DGAT1 (0.44) DGAT1SOAT1KCNH2ADORA2AIDO1
SCHEMBL901631 0.68 CDK9 (0.32) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed