SCHEMBL9021702

SCHEMBL9021702

COC(=O)CCCCCCN1C2CCCC1CC(NC(=O)c1ccc(NC(C)=O)cc1OC)C2

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
CXCR6 O00574 11/20 0.46
DRD2 P14416 1/20 0.46
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021536 1.00 TSHR (0.47) TSHRCXCR6DRD2CYP2D6CYP2C9
SCHEMBL9021905 1.00 TSHR (0.47) TSHRCXCR6DRD2CYP2D6CYP2C9
SCHEMBL9021580 0.93 TSHR (0.47) TSHRCXCR6DRD2CYP2D6CYP2C9
SCHEMBL9021529 0.90 TSHR (0.48) TSHRCXCR6DRD2
SCHEMBL9022056 0.86 TSHR (0.43) TSHRCXCR6
SCHEMBL9022015 0.86 TSHR (0.49) TSHRCXCR6DRD2CYP2D6CYP2C9
SCHEMBL9021726 0.85 DRD2 (0.52) TSHRCXCR6DRD2
SCHEMBL9021985 0.85 DRD2 (0.52) TSHRCXCR6DRD2
SCHEMBL9021950 0.85 DRD2 (0.52) TSHRCXCR6DRD2
SCHEMBL9021718 0.83 OPRK1 (0.50) TSHRCXCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640601-B1 BENZAMIDE DERIVATIVE HOKURIKU PHARMACEUTICAL (JP) 1996-12-04 EP disclosed
US-5500422-A FOR TREATING GASTROINTESTINAL DISEASES HOKURIKU SEIYAKU CO. LTD. (JP) 1996-03-19 US disclosed
US-5395832-A Gastrointestinal disorders HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-07 US disclosed
EP-0640601-A1 BENZAMIDE DERIVATIVE HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-01 EP disclosed