SCHEMBL902192

SCHEMBL902192

O=C(O)C[C@H]1CC[C@H](c2ccc(-c3ccc(-c4nc5cccc(-n6cnnn6)c5[nH]4)cc3)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 0.52
SOAT1 P35610 2/20 0.52
KCNH2 Q12809 2/20 0.40
ADORA2A P29274 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902399 0.80 DGAT1 (0.60) DGAT1SOAT1
SCHEMBL902749 0.78 DGAT1 (0.55) DGAT1SOAT1
SCHEMBL900619 0.77 DGAT1 (0.56) DGAT1SOAT1
SCHEMBL900620 0.77 DGAT1 (0.56) DGAT1SOAT1
SCHEMBL15073265 0.70 DGAT1 (0.58) DGAT1SOAT1
SCHEMBL901499 0.70 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL900018 0.70 DGAT1 (0.55) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902462 0.70 DGAT1 (0.73) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902547 0.69 DGAT1 (0.78) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901149 0.69 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed