SCHEMBL900018

SCHEMBL900018

COc1cccc2nc(-c3ccc(-c4ccc(C5CCC(CC(=O)O)CC5)cc4)cn3)[nH]c12

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.55
SOAT1 P35610 3/20 0.49
KCNH2 Q12809 5/20 0.48
ADORA2A P29274 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901499 0.93 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189208 0.84 S1PR1 (0.42) DGAT1
SCHEMBL901747 0.77 DGAT1 (0.70) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902393 0.77 DGAT1 (0.42) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189566 0.76 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902399 0.76 DGAT1 (0.60) DGAT1SOAT1
SCHEMBL901149 0.75 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189192 0.75 DGAT1 (0.65) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902749 0.74 DGAT1 (0.55) DGAT1SOAT1
SCHEMBL181011 0.73 DGAT1 (0.49) DGAT1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed