SCHEMBL9023871

SCHEMBL9023871

Clc1ccc(Cn2cnc(CCc3ccccc3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.44
HPGDS O60760 1/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2A6 P11509 2/20 0.43
CYP2B6 P20813 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2E1 P05181 1/20 0.43
PHF8 Q9UPP1 2/20 0.42
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
CYP19A1 P11511 3/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6952807 0.86 SIGMAR1 (0.45) SIGMAR1HPGDSCYP3A4CYP2D6CYP2A6
SCHEMBL20457833 0.86 HPGDS (0.40) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6
SCHEMBL9641996 0.83 CNR1 (0.39) SIGMAR1HPGDSCYP3A4CYP2D6CYP2A6
SCHEMBL27548657 0.80 CYP2C9 (0.47) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6
SCHEMBL6896976 0.80 HPGDS (0.50) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6
SCHEMBL10269258 0.80 CYP19A1 (0.54) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6
SCHEMBL6955809 0.79 HPGDS (0.39) SIGMAR1HPGDSCYP3A4CYP2D6CYP2A6
Hydrochloric Acid SCHEMBL7878223 0.78 TDP1 (0.49) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6
SCHEMBL30741761 0.77 HPGDS (0.50) SIGMAR1HPGDSCYP3A4CYP2D6CYP2A6
SCHEMBL28417084 0.77 HPGDS (0.50) HPGDSCYP3A4CYP2D6CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729459-A1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 1996-09-04 EP disclosed
WO-1995014007-A1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 1995-05-26 WO disclosed