SCHEMBL9024153

SCHEMBL9024153

COc1ccc(CCC2c3c(cc(OC)c(OC)c3O)CCN2C=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 4/20 0.56
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
MTNR1A P48039 1/20 0.44
PDE4D Q08499 7/20 0.42
PDE4A P27815 3/20 0.42
PDE4B Q07343 3/20 0.42
PDE4C Q08493 3/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
PDE6C P51160 1/20 0.41
PDE10A Q9Y233 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
NR1I2 O75469 1/20 0.41
MAOA P21397 1/20 0.41
PTGS2 P35354 1/20 0.41
OPRK1 P41145 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024220 0.90 BCHE (0.54) MTNR1BBCHEACHEMTNR1APDE4D
SCHEMBL9025038 0.83 MTNR1B (0.44) MTNR1BBCHEACHEMTNR1APDE4D
SCHEMBL9024245 0.83 LMNA (0.52) MTNR1BBCHEACHEMTNR1APDE4D
SCHEMBL9024298 0.82 HCRTR1 (0.49) MTNR1BBCHEACHEMTNR1APDE4D
SCHEMBL9025276 0.82 PDE4D (0.51) MTNR1BBCHEACHEMTNR1APDE4D
SCHEMBL9426824 0.81 MTNR1B (0.48) MTNR1BMTNR1APDE4D
SCHEMBL9025364 0.78 MTNR1B (0.50) MTNR1BMTNR1APDE4DPDE4APDE4B
SCHEMBL8982863 0.77 BCHE (0.74) BCHEACHEMAPK1CYP2D6
SCHEMBL9024940 0.76 HCRTR2 (0.49) MTNR1BMTNR1APDE4DMAPK1
SCHEMBL8982764 0.74 TBXA2R (0.49) BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501693-B1 Isoquinoline derivatives BANYU PHARMA CO LTD (JP) 1996-08-28 EP disclosed
US-5362736-A Alkoxy derivatives for cardiovascular disorders BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-11-08 US disclosed
EP-0501693-A1 Isoquinoline derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-09-02 EP disclosed