SCHEMBL9024940

SCHEMBL9024940

COc1cc2c(c(O)c1OC)C(Cc1cccnc1)N(C=O)CC2

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.49
HCRTR1 O43613 1/20 0.49
MTNR1B P49286 2/20 0.46
MTNR1A P48039 1/20 0.44
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PDE4D Q08499 5/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CREBBP Q92793 1/20 0.40
POLB P06746 1/20 0.39
TBXA2R P21731 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024298 0.86 HCRTR1 (0.49) HCRTR2HCRTR1MTNR1BMTNR1APDE4D
SCHEMBL9426824 0.85 MTNR1B (0.48) MTNR1BMTNR1AALDH1A1KDM4EHSD17B10
SCHEMBL9024245 0.84 LMNA (0.52) HCRTR2HCRTR1MTNR1BMTNR1AALDH1A1
SCHEMBL9024220 0.84 BCHE (0.54) HCRTR1MTNR1BMTNR1AALDH1A1KDM4E
SCHEMBL9025038 0.82 MTNR1B (0.44) HCRTR1MTNR1BMTNR1APDE4DTBXA2R
SCHEMBL9025364 0.82 MTNR1B (0.50) MTNR1BMTNR1APDE4D
SCHEMBL9025276 0.78 PDE4D (0.51) MTNR1BMTNR1APDE4D
SCHEMBL9024153 0.76 MTNR1B (0.56) MTNR1BMTNR1AMAPK1PDE4D
SCHEMBL8982857 0.76 TBXA2R (0.54) KDM4ETBXA2R
SCHEMBL21255953 0.71 MTNR1B (0.69) MTNR1BMTNR1APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501693-B1 Isoquinoline derivatives BANYU PHARMA CO LTD (JP) 1996-08-28 EP disclosed
US-5362736-A Alkoxy derivatives for cardiovascular disorders BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-11-08 US disclosed
EP-0501693-A1 Isoquinoline derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-09-02 EP disclosed