SCHEMBL9024249

SCHEMBL9024249

O=C(O)c1ccccc1-n1nc(C(=O)O)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
TSHR P16473 2/20 0.54
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
MYC P01106 3/20 0.47
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
SCN9A Q15858 2/20 0.44
STAT1 P42224 2/20 0.44
ALOX15 P16050 1/20 0.44
RORC P51449 2/20 0.43
BCL2 P10415 1/20 0.43
NR4A1 P22736 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17782553 0.85 BCL2 (0.59) ALDH1A1TSHRMAPTHTTMYC
SCHEMBL9023741 0.83 TSHR (0.72) ALDH1A1TSHRMAPTHTTMYC
SCHEMBL17782595 0.83 ELANE (0.59) TSHRPOLBAPEX1TDP1L3MBTL1
SCHEMBL7421574 0.80 SCN9A (0.58) ALDH1A1TSHRMAPTHTTSCN9A
SCHEMBL17782667 0.79 BCL2 (0.62) ALDH1A1TSHRMAPTMYCBCL2
SCHEMBL4056138 0.77 CYP1A2 (0.42) ALDH1A1TSHRSCN9ASTAT1RORC
SCHEMBL30572213 0.76 CYP1A2 (0.60) ALDH1A1TSHRSTAT1RORCCYP1A2
SCHEMBL9484257 0.76 CYP1A2 (0.60) ALDH1A1TSHRSTAT1RORCCYP1A2
SCHEMBL9025523 0.76 RORC (0.56) ALDH1A1CA12CA9SCN9ASTAT1
SCHEMBL16207551 0.74 TSHR (0.72) ALDH1A1TSHRMAPTHTTMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347749-B1 Pyrazoloacridone derivatives with anti-tumoral activity KYOWA HAKKO KOGYO KK (JP) 1996-04-24 EP disclosed
US-5079358-A Humans; leukemia KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-01-07 US disclosed
EP-0347749-A2 Pyrazoloacridone derivatives with anti-tumoral activity KYOWA HAKKO KOGYO CO., LTD. (JP) 1989-12-27 EP disclosed