SCHEMBL9024372

SCHEMBL9024372

O=C(O)OC1CCN(C(=O)N2CCN(c3ccncc3)CC2)CC1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.59
ITGA2B P08514 11/20 0.59
HRH3 Q9Y5N1 2/20 0.56
AKR1C3 P42330 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
TRPV1 Q8NER1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9023640 0.86 HRH3 (0.59) ITGB3ITGA2BHRH3AKR1C3SMN1; SMN2
SCHEMBL16599286 0.82 AKR1C3 (0.58) ITGB3ITGA2BAKR1C3SMN1; SMN2CYP2C9
SCHEMBL8838123 0.82 ITGB3 (0.70) ITGB3ITGA2BAKR1C3SMN1; SMN2CYP2C9
Hydrochloric Acid SCHEMBL9023636 0.80 ITGB3 (0.64) ITGB3ITGA2BHRH3
SCHEMBL8838202 0.79 AKR1C3 (0.54) ITGB3ITGA2BAKR1C3SMN1; SMN2CYP2C9
SCHEMBL9023984 0.79 AKR1C3 (0.48) ITGB3ITGA2BAKR1C3SMN1; SMN2CYP2C9
SCHEMBL28784972 0.77 HRH3 (0.57) ITGB3ITGA2BHRH3CYP2C9CYP2C19
SCHEMBL27471218 0.76 ALDH1A1 (0.66) ITGB3ITGA2BAKR1C3SMN1; SMN2CYP2C9
SCHEMBL8553302 0.76 HRH3 (0.41) ITGB3ITGA2BHRH3
SCHEMBL7401896 0.76 HRH3 (0.62) ITGB3ITGA2BHRH3SMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0718287-A2 Piperazine derivatives, medicaments containing them, their use, and processes for their preparation Dr. Karl Thomae GmbH (DE) 1996-06-26 EP disclosed