SCHEMBL9024375

SCHEMBL9024375

CCS(=O)(=O)c1ccc(-c2oc(C(c3ccccc3)c3ccccc3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.65
PTGS1 P23219 3/20 0.49
TP53 P04637 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
PTGDR2 Q9Y5Y4 2/20 0.40
MAPT P10636 2/20 0.40
THRB P10828 1/20 0.40
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
CCR6 P51684 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PSIP1 O75475 1/20 0.38
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7503544 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL7499074 0.86 PTGS2 (0.62) PTGS2PTGS1PTGDR2
SCHEMBL8549078 0.79 PTGS2 (0.40) PTGS2PTGS1SMN1; SMN2PTGDR2CYP1A2
SCHEMBL9026582 0.79 PTGS2 (0.64) PTGS2PTGS1TP53SMN1; SMN2CYP3A4
SCHEMBL9025662 0.78 PTGS2 (0.59) PTGS2PTGS1TP53SMN1; SMN2MAPT
SCHEMBL8549766 0.76 PTGS2 (0.71) PTGS2PTGS1TP53SMN1; SMN2MAPT
SCHEMBL9025785 0.76 PTGS2 (0.60) PTGS2PTGS1TP53SMN1; SMN2
SCHEMBL7868750 0.76 PTGS2 (0.67) PTGS2PTGS1PTGDR2CYP3A4HPGD
SCHEMBL8558824 0.75 PTGS2 (0.45) PTGS2PTGS1PTGDR2
SCHEMBL9029716 0.73 PTGS2 (0.59) PTGS2PTGS1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699192-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-06 EP claimed
WO-1994027980-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1994-12-08 WO claimed