SCHEMBL9024445

SCHEMBL9024445

Cc1[nH]c(C(C)C)c(/C=C/C#N)c1-c1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
PTGS2 P35354 4/20 0.33
GCGR P47871 4/20 0.33
MLYCD O95822 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
TYMP P19971 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024739 0.75 NR4A2 (0.34) GAAPTGS2GCGR
SCHEMBL9025290 0.72 PTGS2 (0.33) GAAPTGS2GCGR
SCHEMBL10397582 0.70 GCGR (0.40) PTGS2GCGR
SCHEMBL9083836 0.69 GCGR (0.33) GCGR
SCHEMBL9083842 0.69 GCGR (0.33) GCGR
SCHEMBL9024300 0.69 PTGS2 (0.34) PTGS2
SCHEMBL9410843 0.68 GCGR (0.32) GCGR
SCHEMBL9410841 0.68 GCGR (0.32) GCGR
SCHEMBL8855189 0.67 ALDH1A1 (0.34) GCGR
SCHEMBL9085590 0.67 GCGR (0.31) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464845-B1 Pyrrole derivatives SHIONOGI & CO (JP) 1996-06-05 EP disclosed
US-5128366-A Enzyme inhibitors, anticholesterol SHINOGI & CO., LTD. (JP) 1992-07-07 US disclosed
EP-0464845-A1 Pyrrole derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1992-01-08 EP disclosed