SCHEMBL9024497

SCHEMBL9024497

COS(=O)(=O)NC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2NC1=O

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PYGL P06737 5/20 0.46
PYGM P11217 5/20 0.46
RIPK1 Q13546 14/20 0.44
MC4R P32245 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025748 0.81 PYGL (0.47) PYGLPYGMRIPK1
SCHEMBL8329105 0.81 PYGL (0.47) PYGLPYGMRIPK1
SCHEMBL8329558 0.81 PYGL (0.53) PYGLPYGMRIPK1
SCHEMBL9024004 0.79 PYGL (0.47) PYGLPYGMRIPK1
SCHEMBL9025094 0.78 RIPK1 (0.48) PYGLPYGMRIPK1
SCHEMBL7421739 0.78 RIPK1 (0.48) PYGLPYGMRIPK1
SCHEMBL9026043 0.78 RIPK1 (0.48) PYGLPYGMRIPK1
SCHEMBL7792280 0.77 PYGL (0.58) PYGLPYGMRIPK1
SCHEMBL9025264 0.77 RIPK1 (0.47) PYGLPYGMRIPK1
SCHEMBL8331562 0.75 RIPK1 (0.45) PYGLPYGMRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513974-B1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO INC (US) 1996-09-04 EP disclosed
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed