SCHEMBL9026650

SCHEMBL9026650

[O]CCCCCCc1cc(Cl)c(Cl)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.36
ALOX15 P16050 1/20 0.36
ALDH1A1 P00352 2/20 0.35
PTGS2 P35354 2/20 0.32
CYP3A4 P08684 2/20 0.32
HPGD P15428 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PYGL P06737 1/20 0.31
CBS P35520 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10609249 0.79 IGF1R (0.59) IGF1RALOX15ALDH1A1PYGL
SCHEMBL10610096 0.79 IGF1R (0.59) IGF1RALOX15ALDH1A1PYGL
SCHEMBL10606127 0.79 IGF1R (0.59) IGF1RALOX15ALDH1A1PYGL
SCHEMBL8905774 0.79 IGF1R (0.59) IGF1RALOX15ALDH1A1PYGL
SCHEMBL9026661 0.78 IGF1R (0.40) IGF1RALOX15ALDH1A1PTGS2CYP3A4
SCHEMBL9177319 0.78 IGF1R (0.36) IGF1RALOX15ALDH1A1PTGS2CYP3A4
SCHEMBL8861076 0.78 IGF1R (0.36) IGF1RALOX15ALDH1A1PTGS2CYP3A4
SCHEMBL9177322 0.78 PTGS2 (0.55) ALDH1A1PTGS2CYP3A4HSD17B10
SCHEMBL11199961 0.78 CBS (0.39) IGF1RALOX15ALDH1A1CBS
SCHEMBL11199932 0.78 IGF1R (0.33) IGF1RALOX15ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0411150-B1 INDOLE DERIVATIVES, PREPARATION THEREOF, AND DRUG FOR PREVENTING AND TREATING NEPHRITIS CONTAINING SAME OTSUKA PHARMA CO LTD (JP) 1996-11-27 EP disclosed
US-5459142-A Autoimmune disease, atherosclerosis, antiischemic agents and nephritis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-17 US disclosed
EP-0511879-B1 Pyrazine derivatives OTSUKA PHARMA CO LTD (JP) 1995-03-22 EP disclosed
US-5238938-A Nephrosis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-08-24 US disclosed
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed
EP-0411150-A1 INDOLE DERIVATIVES, PREPARATION THEREOF, AND DRUG FOR PREVENTING AND TREATING NEPHRITIS CONTAINING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-02-06 EP disclosed