SCHEMBL9028491

SCHEMBL9028491

COCCn1cc(C(=O)O)c(=O)c2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.63
CHRM1 P11229 1/20 0.62
CNR1 P21554 3/20 0.62
CNR2 P34972 3/20 0.62
ALDH1A1 P00352 2/20 0.57
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6042188 0.90 CNR2 (0.70) LMNACNR1CNR2ALDH1A1MAPT
SCHEMBL9029183 0.85 LMNA (0.68) LMNACHRM1CNR1CNR2
SCHEMBL10656688 0.84 CNR2 (0.76) CNR1CNR2ALDH1A1MAPTTSHR
SCHEMBL10086145 0.83 ALDH1A1 (0.56) LMNACHRM1CNR1CNR2ALDH1A1
SCHEMBL29874516 0.83 LMNA (0.69) LMNACHRM1CNR2
SCHEMBL9026679 0.82 CNR2 (0.74) LMNACNR1CNR2
SCHEMBL90348 0.82 CNR2 (0.71) LMNACNR1CNR2ALDH1A1MAPT
SCHEMBL3450091 0.82 ALDH1A1 (0.46) LMNACHRM1CNR1CNR2ALDH1A1
SCHEMBL4154426 0.82 KDM4E (0.55) LMNACHRM1CNR1CNR2ALDH1A1
SCHEMBL1661468 0.81 LMNA (0.71) LMNACHRM1CNR2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494978-B1 HETEROCYCLIC COMPOUNDS WYETH JOHN & BROTHER LTD (GB) 1996-02-28 EP disclosed
US-5362734-A Certain benzo-quinolizine compounds and derivatives thereof AMERICAN HOME PRODUCTS CORPORATION (US) 1994-11-08 US disclosed
US-5225419-A Antagonist 5-hydroxytryptamine for treatment of nausea or vomiting JOHN WYETH & BROTHER, LIMITED (GB) 1993-07-06 US disclosed
EP-0494978-A1 HETEROCYCLIC COMPOUNDS. WYETH JOHN & BROTHER LTD (GB) 1992-07-22 EP disclosed
US-5096901-A PHARMACOLOGICALLY ACTIVE AMIDES AND ESTERS CONTAINING AN AZABICYCLOALKANE MOIETY JOHN WYETH & BROTHER LIMITED (GB) 1992-03-17 US disclosed
WO-1991005783-A1 HETEROCYCLIC COMPOUNDS JOHN WYETH & BROTHER LIMITED (GB) 1991-05-02 WO disclosed