SCHEMBL9028663

SCHEMBL9028663

CCOc1ccc([C@@]2(CCOS(C)(=O)=O)CCCCN(C(=O)Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)C2)cc1OCC

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTT P42858 1/20 0.37
USP2 O75604 2/20 0.36
CYP3A4 P08684 2/20 0.36
GLA P06280 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
TACR1 P25103 7/20 0.35
SLC6A4 P31645 2/20 0.35
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.35
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
CNR1 P21554 1/20 0.34
HIF1A Q16665 1/20 0.34
TACR2 P21452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026989 0.98 CYP3A4 (0.38) MEN1KMT2AHTTUSP2CYP3A4
SCHEMBL8885684 0.94 TACR1 (0.40) MEN1KMT2AUSP2CYP3A4TACR1
SCHEMBL9028318 0.91 MAPT (0.41) MEN1KMT2AUSP2CYP3A4GLA
SCHEMBL9027943 0.88 TACR1 (0.41) MEN1KMT2AUSP2CYP3A4GLA
SCHEMBL9027536 0.88 MEN1 (0.39) MEN1KMT2AUSP2CYP3A4GLA
SCHEMBL9027646 0.88 TACR2 (0.42) MEN1KMT2ATACR1TACR2
SCHEMBL9027505 0.88 TACR2 (0.42) MEN1KMT2ATACR1TACR2
SCHEMBL9028344 0.87 MEN1 (0.40) MEN1KMT2AUSP2CYP3A4GLA
SCHEMBL9028480 0.87 MEN1 (0.40) MEN1KMT2AUSP2CYP3A4GLA
SCHEMBL9028382 0.87 MEN1 (0.40) MEN1KMT2AUSP2CYP3A4GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed