SCHEMBL9028745

SCHEMBL9028745

CC=C(C)Oc1cc(C(C)C)c(OC(C)=O)c(C(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.38
HTT P42858 2/20 0.37
CYP1A2 P05177 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
PKM P14618 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
ADRA1D P25100 1/20 0.36
HTR2C P28335 1/20 0.36
ADRA1A P35348 1/20 0.36
HRH1 P35367 1/20 0.36
ADRA1B P35368 1/20 0.36
DRD3 P35462 1/20 0.36
OPRK1 P41145 1/20 0.36
CHRNA4 P43681 1/20 0.36
HIF1A Q16665 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TP53 P04637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9029438 0.88 BACE1 (0.47) BACE1HTTPKMSMN1; SMN2KDM4E
SCHEMBL17935193 0.78 CA1 (0.46) BACE1HTTCYP1A2ADRA2ACYP2D6
SCHEMBL9028778 0.77 AKR1B1 (0.38) HTTCYP1A2ADRA2ACYP2D6PKM
SCHEMBL8176820 0.77 FABP3 (0.52) HTTRARGRXRAPPARG
SCHEMBL6768274 0.77 PREP (0.42) BACE1HTTCYP1A2ADRA2ACYP2D6
SCHEMBL9270934 0.76 FNTA (0.42) HTTCYP1A2ADRA2ACYP2D6PKM
SCHEMBL1928602 0.75 GABRA1 (0.40) HTTCYP1A2ADRA2ACYP2D6PKM
SCHEMBL29113877 0.75 HTT (0.38) BACE1HTTCYP1A2ADRA2ACYP2D6
SCHEMBL6767046 0.74 BACE1 (0.40) BACE1SMN1; SMN2KDM4ETP53MAPT
SCHEMBL9090807 0.74 THRA (0.45) BACE1KDM4ELMNAGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445827-B1 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO KK (JP) 1996-09-25 EP disclosed
US-5149834-A Anticholesterol agent and enzyme inhibitors, for curing arteriosclerosis FUJIREBIO INC. (JP) 1992-09-22 US disclosed
EP-0445827-A2 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO INC. (JP) 1991-09-11 EP disclosed