SCHEMBL9028778

SCHEMBL9028778

CC=C(C)Oc1c(O)cc(C(C)C)c(OC(C)=O)c1C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.38
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
HTT P42858 2/20 0.36
GAA P10253 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP1A2 P05177 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2D6 P10635 1/20 0.33
PKM P14618 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1D P25100 1/20 0.33
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767136 0.78 MAPT (0.36) AKR1B1LDHALDHBHTTGAA
SCHEMBL9028745 0.77 BACE1 (0.38) AKR1B1LDHALDHBHTTGAA
SCHEMBL9028770 0.77 RXRA (0.35) AKR1B1LDHALDHBHTTGAA
SCHEMBL6766511 0.71 LDHA (0.33) AKR1B1LDHALDHBHTTGAA
SCHEMBL6768274 0.71 PREP (0.42) AKR1B1LDHALDHBHTTGAA
SCHEMBL5042710 0.69 HTT (0.45) AKR1B1LDHALDHBHTTGAA
SCHEMBL17935193 0.69 CA1 (0.46) HTTCYP1A2ADRA2ACYP2D6PKM
SCHEMBL4469962 0.69 CYP3A4 (0.39) AKR1B1LDHALDHBHTTGAA
SCHEMBL9029438 0.68 BACE1 (0.47) HTTKDM4ETP53MAPTPKM
SCHEMBL8176820 0.68 FABP3 (0.52) HTTRARGRXRAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445827-B1 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO KK (JP) 1996-09-25 EP disclosed
US-5149834-A Anticholesterol agent and enzyme inhibitors, for curing arteriosclerosis FUJIREBIO INC. (JP) 1992-09-22 US disclosed
EP-0445827-A2 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO INC. (JP) 1991-09-11 EP disclosed